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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 10 hits in this display   

TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human beta2 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog recombinant beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by enzyme immuno assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50: >3.20E+3nMAssay Description:Agonist activity at human beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at dog beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human cloned beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50: >3.20E+3nMAssay Description:Agonist activity at human cloned beta-1 adrenergic receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50240563(CHEMBL59765 | ethyl 2-((S)-8-((R)-2-(3-chloropheny...)
Affinity DataEC50:  16nMAssay Description:Agonist activity at human beta3 adrenergic receptor expressed in CHO cells assessed as cAMP accumulation by EIAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed