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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetApoptotic protease-activating factor 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataIC50:  797nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBIMR, San Diego, C...More data for this Ligand-Target Pair
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TargetCaspase-9(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataIC50:  1.37E+3nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBIMR, San Diego, C...More data for this Ligand-Target Pair
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TargetMothers against decapentaplegic homolog 3(Homo sapiens (Human))
Emory University

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataIC50:  1.04E+4nMAssay Description:NIH Molecular Libraries Screening Centers Network [MLSCN] Emory Chemical Biology Discovery Center in MLSCN Assay provider: F.M. Hoffmann, University ...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataIC50:  1.04E+4nMAssay Description:List of compounds to be tested: Compounds that met the active criterion of Z-score is More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetApoptotic protease-activating factor 1(Homo sapiens (Human))
Burnham Center For Chemical Genomics

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataIC50: >1.00E+5nMAssay Description:Data Source: Sanford-Burnham Center for Chemical Genomics (SBCCG) Source Affiliation: Sanford-Burnham Medical Research Institute (SBIMR, San Diego, C...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataEC50:  614nMAssay Description:List of compounds to be tested: Compounds that met the active criterion of Z-score is More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University of Pittsburgh

Curated by PubChem BioAssay
LigandPNGBDBM40316(8-bromo-2,3-dimethyl-4,5-dioxo-1-benzo[e]indolecar...)
Affinity DataEC50:  723nMAssay Description:List of compounds to be tested: Compounds that met the active criterion of Z-score is More data for this Ligand-Target Pair
In DepthDetails PCBioAssay