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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 12 hits in this display   

Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]LSD from 5-HT2B receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  174nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 5A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  457nMAssay Description:Displacement of [3H]LSD from 5-HT5A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 7(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  472nMAssay Description:Displacement of [3H]LSD from 5-HT7A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  714nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  851nMAssay Description:Displacement of [3H]LSD from 5-HT2C receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  3.59E+3nMAssay Description:Displacement of [3H]LSD from 5-HT6 receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi:  8.59E+3nMAssay Description:Displacement of [3H]GR127543 from 5-HT1D receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]GR127543 from 5-HT1B receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]LY278584 from 5-HT3 receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1E(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-5-HT from 5-HT1E receptor (unknown origin) after 1.5 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing

Curated by ChEMBL
LigandPNGBDBM50148833(CHEMBL3770106)
Affinity DataIC50:  27nMAssay Description:Antagonist activity at 5-HT2B receptor (unknown origin) expressed in CHO-K1 cells assessed as calcium flux after 60 mins by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed