Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 12 hits in this display
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: <10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: <10nMAssay Description:FGFR1, FGFR2, and FGFR4 are measured under equivalent conditions with the following changes in enzyme and ATP concentrations: FGFR1, 0.02 nM and 210 ...More data for this Ligand-Target Pair
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: 20nMAssay Description:FGFR1, FGFR2, and FGFR4 are measured under equivalent conditions with the following changes in enzyme and ATP concentrations: FGFR1, 0.02 nM and 210 ...More data for this Ligand-Target Pair
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
BDBM262071(3-(2,6-difluoro-3,5- dimethoxyphenyl)-7-(1,3- dime...)
IC50: 20nMAssay Description:FGFR1, FGFR2, and FGFR4 are measured under equivalent conditions with the following changes in enzyme and ATP concentrations: FGFR1, 0.02 nM and 210 ...More data for this Ligand-Target Pair