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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Mast/stem cell growth factor receptor Kit [D816V]
(Homo sapiens (Human))
Plexxikon
US Patent
Ligand
BDBM342294
(4-[4-[5-(3-ethoxy-4-methyl-phenyl)-4- methyl-1H-im...)
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Affinity Data
Ki: 500nM
Assay Description:
The c-kit mutant D816V (or kinase domain thereof) is an active kinase in AlphaScreen. IC50 values are determined with respect to inhibition of c-Kit ...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Plexxikon
US Patent
Ligand
BDBM342294
(4-[4-[5-(3-ethoxy-4-methyl-phenyl)-4- methyl-1H-im...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 500nM
Assay Description:
Assays for biochemical cell-based activity of c-kit kinase are known in the art, for example, as described in U.S. Pat. Nos. 7,498,342 and 7,846,941,...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI