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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50205338(CHEMBL3948237)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of GST/His-tagged human KEAP1 (321 to 609 residues) interaction with phosphorylated p62 expressed in Escherichia coli cells by fluorescenc...More data for this Ligand-Target Pair
TargetKelch-like ECH-associated protein 1(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50205338(CHEMBL3948237)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of KEAP1/Nrf2 (unknown origin) protein-protein interactionMore data for this Ligand-Target Pair
TargetNuclear factor erythroid 2-related factor 2(Homo sapiens (Human))
Keio University

Curated by ChEMBL
LigandPNGBDBM50205338(CHEMBL3948237)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of recombinant GST-His-tagged Keap1-DC domain (321 to 609 residues) (unknown origin) expressed in Escherichia coli/FAM-labeled Nrf2 (unkno...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed