Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL

LigandBDBM50508145(CHEMBL4450146)Copy SMILESCopy InChI

Affinity DataIC50:  30nMAssay Description:Antagonist activity at recombinant human PPARdelta assessed as inhibition of GW0742-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Inception Sciences

Curated by ChEMBL

LigandBDBM50508145(CHEMBL4450146)Copy SMILESCopy InChI

Affinity DataIC50:  216nMAssay Description:Antagonist activity at recombinant human PPARalpha assessed as inhibition of GW7647-induced receptor activation after overnight incubation by cell-ba...More data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI