Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetD(2) dopamine receptor(Homo sapiens (Human))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  22nMAssay Description:In vitro binding affinity towards D2 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Mus musculus (Mouse))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  22nMAssay Description:Binding affinity of the compound towards Dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  27nMAssay Description:In vitro inhibition of [3H]8-OH-DPAT binding to 5-hydroxytryptamine 1A receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  27nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 1A receptor was determined using radioligand [3H]-8-OH-DPATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Mus musculus (Mouse))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi:  27nMAssay Description:Binding affinity of the compound towards 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 2A receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mus musculus (Mouse))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-HT4 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro inhibition of [3H]prazosin binding to Alpha-1 adrenergic receptor in rat cerebral cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Universidad Complutense

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL1204203 | CHEMBL416266 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:In vitro binding affinity towards 5-hydroxytryptamine 3 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed