Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetFibroblast growth factor receptor 2(Homo sapiens (Human))
Incyte

US Patent

LigandBDBM592107(US11566028, Example 46)Copy SMILESCopy InChI

Affinity DataIC50: <10nMMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetFibroblast growth factor receptor 3(Homo sapiens (Human))
Incyte

US Patent

LigandBDBM592107(US11566028, Example 46)Copy SMILESCopy InChI

Affinity DataIC50:  20nMAssay Description:The inhibitor potency of the exemplified compounds was determined in an enzyme discontinuous assay that measures peptide phosphorylation using FRET m...More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetFibroblast growth factor receptor 1(Homo sapiens (Human))
Incyte

US Patent

LigandBDBM592107(US11566028, Example 46)Copy SMILESCopy InChI

Affinity DataIC50:  20nMMore data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI

TargetFibroblast growth factor receptor 4(Homo sapiens (Human))
Incyte

US Patent

LigandBDBM592107(US11566028, Example 46)Copy SMILESCopy InChI

Affinity DataIC50: >200nMMore data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
DrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails US Patent
Copy BDB DOI