Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 18 hits in this display
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
BDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
BDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
IC50: 64nMpH: 7.2 T: 2°CAssay Description:The MLK kinase assays were performed by using the Millipore multiscreen trichloroacetic acid (TCA) in-plate format. The inhibition curves were genera...More data for this Ligand-Target Pair
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
IC50: >1.00E+3nMAssay Description:Ability to inhibit human trk A tyrosine kinase expressed in baculovirus using ELISA based enzyme assay was determinedMore data for this Ligand-Target Pair
BDBM50058332(CHEMBL299496 | methyl 10,23-di(ethylsulfanylmethyl...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)
BDBM24942(CEP-1347 | CHEMBL290352 | methyl (15S,16R,18R)-10,...)