Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetTranscription factor 4(Homo sapiens)
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589362(CHEMBL5181203)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of His-tagged beta-catenin (134 to 668 residues)/CM-5 sensor chip immobilized N-terminal GST-tagged TCF4 interaction (unknown origin) prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetCatenin beta-1(Homo sapiens (Human))
Vu University Amsterdam

Curated by ChEMBL
LigandPNGBDBM50589362(CHEMBL5181203)
Affinity DataKd:  5.80E+5nMAssay Description:Binding affinity to CM-5 sensor chip immobilized His-tagged beta-catenin (134 to 668 residues) (unknown origin) expressed in Escherichia coli BL21 as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed