Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50256510(CHEMBL500977 | N-(5-ethyl-1,3,4-thiadiazol-2-yl)su...)
Ki: 950nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 2 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256510(CHEMBL500977 | N-(5-ethyl-1,3,4-thiadiazol-2-yl)su...)
Ki: 7.01E+3nMAssay Description:Inhibition of human recombinant cytosolic carbonic anhydrase 1 pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256510(CHEMBL500977 | N-(5-ethyl-1,3,4-thiadiazol-2-yl)su...)
Ki: 8.64E+3nMAssay Description:Inhibition of truncated human cloned membrane-associated carbonic anhydrase 4 preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256510(CHEMBL500977 | N-(5-ethyl-1,3,4-thiadiazol-2-yl)su...)
Ki: 1.87E+4nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5A pre-incubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair
BDBM50256510(CHEMBL500977 | N-(5-ethyl-1,3,4-thiadiazol-2-yl)su...)
Ki: 6.30E+4nMAssay Description:Inhibition of full length human recombinant mitochondrial carbonic anhydrase 5B preincubated for 15 mins by stopped-flow CO2 hydration assayMore data for this Ligand-Target Pair