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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Cyclin-H/Cyclin-dependent kinase 7
(Homo sapiens (Human))
Dana-Farber Cancer Institute
US Patent
Ligand
BDBM464109
(US10787436, Compound I-52 | US10787436, Compound I...)
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Affinity Data
IC50: <100nM
Assay Description:
In vitro kinase assays with immunoprecipitated proteins (or recombinant CAK complexes) were performed as follows. Kinase reactions were performed in ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Cyclin-H/Cyclin-dependent kinase 7
(Homo sapiens (Human))
Dana-Farber Cancer Institute
US Patent
Ligand
BDBM464109
(US10787436, Compound I-52 | US10787436, Compound I...)
Copy SMILES
Copy InChI
Affinity Data
IC50: <100nM
Assay Description:
In vitro kinase assays with immunoprecipitated proteins (or recombinant CAK complexes) were performed as follows. Kinase reactions were performed in ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Cyclin-dependent kinase 5 activator 1 [99-307]
(Homo sapiens (Human))
Dana-Farber Cancer Institute
US Patent
Ligand
BDBM464109
(US10787436, Compound I-52 | US10787436, Compound I...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 550nM
Assay Description:
In vitro kinase assays with immunoprecipitated proteins (or recombinant CAK complexes) were performed as follows. Kinase reactions were performed in ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
Dana-Farber Cancer Institute
US Patent
Ligand
BDBM464109
(US10787436, Compound I-52 | US10787436, Compound I...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 550nM
Assay Description:
In vitro kinase assays with immunoprecipitated proteins (or recombinant CAK complexes) were performed as follows. Kinase reactions were performed in ...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI