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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetHistamine H1 receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50:  17nMAssay Description:Binding affinity against Histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50:  912nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(4) dopamine receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Alpha-3A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against 5-HT1D receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against 5-HT2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against 5-HT1A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2LMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Janssen-Cilag

Curated by ChEMBL
LigandPNGBDBM50421590(CHEMBL331188)
Affinity DataIC50: <1.00E+3nMAssay Description:Binding affinity against Alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed