Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetMuscarinic acetylcholine receptor M4(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.5nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.70nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  1.90nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataKi:  27nMAssay Description:Antimuscurinic potency and subset specificity of the compound was characterised by its inhibition of the [3H]-NMS Binding to Muscarinic acetylcholine...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPancreatic alpha-amylase(Rattus norvegicus)
Institute of Research

Curated by ChEMBL
LigandPNGBDBM50005681(2-Cyclohexyl-2-phenyl-propionic acid 3-dimethylami...)
Affinity DataIC50:  10nMAssay Description:Inhibition of the release of Alpha-amylase from rat pancreatic acinar cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed