Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Norwegian University Of Science And Technology

Curated by ChEMBL

LigandBDBM50449656(CHEMBL4159505)Copy SMILESCopy InChI

Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at GAL4-DBD fused human RORgamma LBD expressed in HEK293 cells after 18 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetLuciferin 4-monooxygenase(Photinus pyralis)
Norwegian University Of Science And Technology

Curated by ChEMBL

LigandBDBM50449656(CHEMBL4159505)Copy SMILESCopy InChI

Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of firefly luciferase activity expressed in HEK293 cells after 18 hrs by luminescence assayMore data for this Ligand-Target Pair

Target InfoPDBMMDB
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI