Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetP2Y purinoceptor 1(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi:  17nMAssay Description:Binding affinity to human P2Y1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi: >1.50E+4nMAssay Description:Binding affinity to factor-7a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi: >2.50E+4nMAssay Description:Binding affinity to factor-10a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 12(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity to P2Y12 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 2(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi: >3.00E+4nMAssay Description:Binding affinity to P2Y2 receptor (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor XI(Homo sapiens (Human))
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50433784(CHEMBL2381898)
Affinity DataKi: >5.50E+4nMAssay Description:Binding affinity to factor-11a (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed