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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetCathepsin K(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50402198(CHEMBL2203960)
Affinity DataKi:  880nMAssay Description:Inhibition of human recombinant cathepsin K using Z-Leu-Arg-AMC as substrate after 10 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50402198(CHEMBL2203960)
Affinity DataKi:  6.60E+3nMAssay Description:Inhibition of human recombinant cathepsin S using Z-Phe-Arg-pNA as substrate after 10 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
University Of Bonn

Curated by ChEMBL
LigandPNGBDBM50402198(CHEMBL2203960)
Affinity DataKi: >4.00E+4nMAssay Description:Inhibition of human recombinant cathepsin B using Z-Arg-Arg-pNA as substrate after 10 mins by fluorimetric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed