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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Histamine H3 receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
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Affinity Data
Ki: 37nM
Assay Description:
Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
Copy SMILES
Copy InChI
Affinity Data
Ki: 37.1nM
Assay Description:
Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Rattus norvegicus (rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
Copy SMILES
Copy InChI
Affinity Data
Ki: 214nM
Assay Description:
Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membrane
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Rattus norvegicus (rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
Copy SMILES
Copy InChI
Affinity Data
Ki: 214nM
Assay Description:
Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
Copy SMILES
Copy InChI
Affinity Data
Ki: 6.46E+3nM
Assay Description:
Displacement of [3H]RAMHA from human histamine H4 receptor expressed in SK-N-MC cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Acetylcholinesterase
(Rattus norvegicus (rat))
Universit£
Curated by
ChEMBL
Ligand
BDBM50412459
(CHEMBL212775)
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Affinity Data
IC50: 1.66E+3nM
Assay Description:
Inhibition of acetylcholinesterase in Wistar rat brain homogenate by Ellman's method
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI