Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataKi:  37nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor transfected in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataKi:  37.1nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataKi:  214nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in rat brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataKi:  6.46E+3nMAssay Description:Displacement of [3H]RAMHA from human histamine H4 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Rattus norvegicus (rat))
Universit£

Curated by ChEMBL
LigandPNGBDBM50412459(CHEMBL212775)
Affinity DataIC50:  1.66E+3nMAssay Description:Inhibition of acetylcholinesterase in Wistar rat brain homogenate by Ellman's methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed