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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Mitobridge
US Patent
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
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Affinity Data
EC50: 694nM
Assay Description:
Medium including test compound was aspirated and washed with PBS. 50 μl PBS including 1 mM Mg++ and Ca++ were then added to each well. The lucif...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
PPAR delta protein
(Rattus norvegicus (Rat))
Mitobridge
US Patent
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 694nM
Assay Description:
Medium including test compound was aspirated and washed with PBS. 50 μl PBS including 1 mM Mg++ and Ca++ were then added to each well. The lucif...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/TrEMBL
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor gamma
(Homo sapiens (Human))
Mitobridge
Curated by
ChEMBL
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
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Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Activation of human PPARgamma LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor alpha
(Homo sapiens (Human))
Mitobridge
Curated by
ChEMBL
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Activation of human PPARalpha LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Mitobridge
US Patent
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 690nM
Assay Description:
Activation of human PPARdelta LBD expressed in CHO-K1 cells by beta galactosidase enzyme fragment complement based fluorescence assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Peroxisome proliferator-activated receptor delta
(Homo sapiens (Human))
Mitobridge
US Patent
Ligand
BDBM323597
((E)-6-(2-((4-(furan-2-yl)-N-methylbenzamido)methyl...)
Copy SMILES
Copy InChI
Affinity Data
EC50: >1.00E+4nM
Assay Description:
Transactivation of yeast GAL4 DNA binding domain-fused PPARdelta LBD (unknown origin) expressed in CV-1 cells after 24 hrs by luciferase reporter gen...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI