Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
Ki: 88nMAssay Description:Binding affinity to human XIAP linker BIR2-BIR3 domain expressed in Escherichia coli BL21(DE3) cells by fluorescence polarization-based assayMore data for this Ligand-Target Pair
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)
IC50: 280nMAssay Description:Competitive inhibition of human XIAP linker BIR2-BIR3 domain expressed in Escherichia coli BL21(DE3) cells by fluorescence polarization-based assayMore data for this Ligand-Target Pair
BDBM50343513((3S,6S,10aS)-6-((S)-2-acetamido-3-(1H-indol-3-yl)p...)