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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252702(CHEMBL521656 | N-Methyl-ETAV)
Affinity DataKi:  8.90E+3nMAssay Description:Binding affinity to human PSD95 domain PDZ2 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50339563((3S,6S,9S,12S)-3-(2-carboxyethyl)-6-((R)-1-hydroxy...)
Affinity DataKi:  9.65E+3nMAssay Description:Inhibition of PSD-95 PDZ2 domain by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252702(CHEMBL521656 | N-Methyl-ETAV)
Affinity DataKi:  1.10E+4nMAssay Description:Binding affinity to human PSD95 domain PDZ1 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDisks large homolog 4(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50252702(CHEMBL521656 | N-Methyl-ETAV)
Affinity DataKi:  7.80E+4nMAssay Description:Binding affinity to human PSD95 domain PDZ3 expressed in Escherichia coli BL21-DE3 by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed