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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of North Texas Health Science Center

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataKi:  598nMAssay Description:Displacement of [3H]methylspiperone from human cloned 5HT2A receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataKi:  3.03E+3nMAssay Description:Displacement of [3H]GR65630 from human recombinant 5HT3 receptor expressed in HEKT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of North Texas Health Science Center

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataKi:  1.45E+4nMAssay Description:Displacement of [3H]mesulergine from human cloned 5HT2C receptor expressed in HEK293 cells after 90 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human recombinant MAO-A using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Mississippi

Curated by ChEMBL
LigandPNGBDBM50321885((E)-5-((1H-Indol-3yl)methylene)-2-imino-1,3-dimeth...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human recombinant MAO-B using kynuramine as substrate preincubated with compound for 15 mins measured after 20 mins by fluorometric ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed