Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM242959(US9422277, 22 | US9422277, 84)
BDBM242959(US9422277, 22 | US9422277, 84)
Ki: 13.0nM ΔG°: -45.8kJ/molepH: 5.0 T: 2°CAssay Description:Inhibitor compounds, prepared at 3× the desired final concentration in 1×BACE assay buffer (20 mM sodium acetate pH 5.0, 10% glycerol, 0....More data for this Ligand-Target Pair
BDBM242959(US9422277, 22 | US9422277, 84)
BDBM242959(US9422277, 22 | US9422277, 84)
Ki: 102nM ΔG°: -40.6kJ/molepH: 5.0 T: 2°CAssay Description:Varying concentrations of inhibitors at 3× the final desired concentration in a volume of 10 ul are preincubated with purified human BACE1 cata...More data for this Ligand-Target Pair