Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 4 hits in this display
BDBM242225(US9416129, 3 | US9416129, 5)
BDBM242225(US9416129, 3 | US9416129, 5)
Ki: 7.5nM ΔG°: -47.2kJ/molepH: 5.0 T: 2°CAssay Description:Varying concentrations of inhibitors at 3× the final desired concentration in a volume of 10 μl are preincubated with purified human BACE1 c...More data for this Ligand-Target Pair
BDBM242225(US9416129, 3 | US9416129, 5)
BDBM242225(US9416129, 3 | US9416129, 5)
Ki: 25.9nM ΔG°: -44.0kJ/molepH: 5.0 T: 2°CAssay Description:Inhibitor compounds, prepared at 3× the desired final concentration in 1×BACE assay buffer (20 mM sodium acetate pH 5.0, 10% glycerol, 0....More data for this Ligand-Target Pair