Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM221537(US9303045, 22 | US9695195, 22)
BDBM221584(US9303045, 70 | US9695195, 70)
IC50: 1.13nMT: 2°CAssay Description:The 5HT3 antagonist activity of the compounds of the invention was determined by measuring the ability of the compounds to inhibit the calcium flux a...More data for this Ligand-Target Pair
BDBM221584(US9303045, 70 | US9695195, 70)
BDBM221537(US9303045, 22 | US9695195, 22)
IC50: 1.13nMT: 2°CAssay Description:The 5HT3 antagonist activity of the compounds of the invention was determined by measuring the ability of the compounds to inhibit the calcium flux a...More data for this Ligand-Target Pair
BDBM221594(US9303045, 81 | US9695195, 81)
IC50: 1.44nMT: 2°CAssay Description:The 5HT3 antagonist activity of the compounds of the invention was determined by measuring the ability of the compounds to inhibit the calcium flux a...More data for this Ligand-Target Pair
BDBM221594(US9303045, 81 | US9695195, 81)
IC50: 1.44nMT: 2°CAssay Description:The 5HT3 antagonist activity of the compounds of the invention was determined by measuring the ability of the compounds to inhibit the calcium flux a...More data for this Ligand-Target Pair