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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50133009
((4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-...)
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Affinity Data
Ki: 32nM
Assay Description:
Displacement of [3H]histamine from recombinant human histamine H4 receptor in SK-N-MC cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50133009
((4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 32nM
Assay Description:
Displacement of [3H]- histamine from the recombinant human histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50133009
((4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.19E+7nM
Assay Description:
Antagonist activity at Homo sapiens (human) histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI
Target
Histamine H4 receptor
(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research And Development
Curated by
ChEMBL
Ligand
BDBM50133009
((4-Bromo-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 3.20E+7nM
Assay Description:
Antagonist activity at Homo sapiens (human) histamine H4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
Copy BDB DOI