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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Johann Wolfgang Goethe University
Curated by
ChEMBL
Ligand
BDBM50304501
(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
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Affinity Data
Ki: 290nM
Assay Description:
Displacement of [3H]histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai2 and Gbeta1gamma2
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
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CHEMBL
PC cid
PC sid
Patents
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In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Johann Wolfgang Goethe University
Curated by
ChEMBL
Ligand
BDBM50304501
(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 530nM
Assay Description:
Displacement of [3H]Histamine from human histamine H4 receptor expressed in Sf9 cells co-expressing Galphai/o and Gbeta1gamma
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Histamine H3 receptor
(Homo sapiens (Human))
Ku Leuven
Curated by
ChEMBL
Ligand
BDBM50304501
(6-(4-Methylpiperazin-1-yl)pyrimidine-2,4-diamine |...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.08E+3nM
Assay Description:
Displacement of [3H]Nalpha-methylhistamine from human histamine H3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI