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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 13 hits in this display   

TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  21nMAssay Description:Inhibition of human Cathepsin C in human U-937 cells using H-Gly-Phe-AFC as substrate pretreated for 60 mins followed by substrate addition incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  24nMAssay Description:Inhibition of human Cathepsin C in human THP-1 cells using H-Gly-Phe-AFC as substrate pretreated for 60 mins followed by substrate addition incubated...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  57nMAssay Description:Inhibition of human recombinant Cathepsin C using H-Gly-Arg-AMC as substrate pretreated for 30 mins followed by substrate addition and incubated for ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDipeptidyl peptidase 1(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  57nMAssay Description:Inhibition of human recombinant Cathepsin C using H-Gly-Arg-AMC as substrate pretreated for 30 mins followed by substrate addition incubated for 60 m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  7.13E+3nMAssay Description:Inhibition of recombinant human CYP3A4More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Cathepsin S (unknown origin) using MCA-Arg-Pro-Lys-Pro-Val-Glu-NVAL-Trp-Arg-Lys-(DNP)-NH2 as substrate pretreated for 60 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProcathepsin L(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Cathepsin L (unknown origin) using Z-Leu-Arg-AMC as substrate pretreated for 60 mins followed by substrate addition incubated for 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin B(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Cathepsin B (unknown origin) using Z-Leu-Arg-AMC as substrate pretreated for 60 mins followed by substrate addition incubated for 30 mi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCathepsin K(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Cathepsin K (unknown origin) using MCA-Arg-Pro-Lys-Pro-Val-Glu-NVAL-Trp-Arg-Lys-(DNP)-NH2 as substrate pretreated for 60 mins followed ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant human CYP1A2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  2.54E+4nMAssay Description:Inhibition of recombinant human CYP2D6More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50:  4.94E+4nMAssay Description:Inhibition of recombinant human CYP2C9More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50573801(CHEMBL4859234)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of recombinant human CYP2C19More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed