Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 17 hits in this display   

TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50:  4.93E+3nMAssay Description:Inhibition of SIRT6 (unknown origin) using Ac-RYQK(Ac)-AMC as substrate by Fluor de Lys assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 3(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC10 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of SIRT3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 11(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC11 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 6(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC6 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC7 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of HDAC9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to SIRT6 (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50544037(CHEMBL1370863)
Affinity DataKd:  9.76E+3nMAssay Description:Binding affinity to SIRT6 (unknown origin) by surface plasmon resonance assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed