Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetHistone deacetylase 2(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: <200nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 1(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: <200nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 2(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: <200nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50:  2.55E+4nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 6(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: >5.00E+4nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 3(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: >5.00E+4nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone deacetylase 8(Homo sapiens (Human))
Medibiofarma

US Patent
LigandPNGBDBM535861(N-(3-amino-6-(4-fluorophenyl)pyridin-2-yl)-6-(4-me...)
Affinity DataIC50: >5.00E+4nMAssay Description:The inhibitory activities of compounds of present invention were determined using biochemical HDAC assays (Reaction Biology Corp. biochemical assay s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent