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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Cancer Therapeutics Crc
US Patent
Ligand
BDBM155530
(US9012461, 6)
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Affinity Data
IC50: 4.20nM
pH: 7.4
Assay Description:
A biotin labeled peptide is used as substrate (amino acid sequence: Biotin-Glu-Gly-Pro-Trp-Leu-Glu-Glu-Glu-Glu-Glu-Ala-Tyr-Gly-Trp-Met-Asp-Phe-NH2)1S...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Cancer Therapeutics Crc
US Patent
Ligand
BDBM155530
(US9012461, 6)
Copy SMILES
Copy InChI
Affinity Data
IC50: 52nM
pH: 7.0
Assay Description:
Compounds of the invention may be tested for in vitro activity in the following assay: A biotin labeled peptide is used as substrate (amino acid sequ...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Cancer Therapeutics Crc
US Patent
Ligand
BDBM155530
(US9012461, 6)
Copy SMILES
Copy InChI
Affinity Data
Kd: 6.30nM
pH: 7.4 T: 2°C
Assay Description:
Binding parameters of compounds were determined using a Biacore S51 sensor. An anti-GST antibody was immobilized onto a CM5 chip by primary amine-cou...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI