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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM189350
(3-((4-Amino-6-(4-methylpiperazin-1-yl)-1,3,5-triaz...)
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Affinity Data
Ki: 1.46E+4nM
Assay Description:
Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Universit£
Curated by
ChEMBL
Ligand
BDBM189350
(3-((4-Amino-6-(4-methylpiperazin-1-yl)-1,3,5-triaz...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 1.46E+4nM ΔG°: -25.7kJ/mole
pH: 7.4 T: 2°C
Assay Description:
Prior to the experiments, cell membranes were sedimented by a 10 min centrifugation at 4 °C and 16 0009x g and resuspended in binding buffer (12...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
Article
PubMed
Copy BDB DOI