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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189350(3-((4-Amino-6-(4-methylpiperazin-1-yl)-1,3,5-triaz...)
Affinity DataKi:  1.46E+4nMAssay Description:Displacement of [3H]histamine from human H4R expressed in Sf9 cell membranes co-expressed with G protein Gai2 and Gb1gamma2 incubated for 60 mins by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM189350(3-((4-Amino-6-(4-methylpiperazin-1-yl)-1,3,5-triaz...)
Affinity DataKi:  1.46E+4nM ΔG°:  -25.7kJ/molepH: 7.4 T: 2°CAssay Description:Prior to the experiments, cell membranes were sedimented by a 10 min centrifugation at 4 °C and 16 0009x g and resuspended in binding buffer (12...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed