Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 8 hits in this display
BDBM123101(US11312693, Example 5 | US8735395, 5)
BDBM123101(US11312693, Example 5 | US8735395, 5)
BDBM123101(US11312693, Example 5 | US8735395, 5)
Ki: 1.17E+3nMpH: 7.0Assay Description:Standard assay conditions for the determination of kinetic constants used a fluorogenic peptide substrate, typically H-D-Ala-Leu-Lys-AMC, and were de...More data for this Ligand-Target Pair
BDBM123101(US11312693, Example 5 | US8735395, 5)
Ki: 2.90E+3nMAssay Description:The assay uses baculovirus-expressed human cathepsin S and the boc-Val-Leu-Lys-AMC fluorescent substrate available from Bachem in a 384 well plate fo...More data for this Ligand-Target Pair
BDBM123101(US11312693, Example 5 | US8735395, 5)
Ki: 2.90E+3nMpH: 7.0Assay Description:Standard assay conditions for the determination of kinetic constants used a fluorogenic peptide substrate, typically H-D-Ala-Leu-Lys-AMC, and were de...More data for this Ligand-Target Pair