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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
5-hydroxytryptamine receptor 3A
(RAT)
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by
ChEMBL
Ligand
BDBM50060685
(9-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)
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Affinity Data
Ki: 0.440nM
Assay Description:
Displacement of [3H]LY278584 from 5HT3 receptor in rat cortical homogenate
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
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Article
PubMed
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Target
5-hydroxytryptamine receptor 3A/3B
(Rattus norvegicus)
Universit£
Curated by
ChEMBL
Ligand
BDBM50060685
(9-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)
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Affinity Data
IC50: 0.440nM
Assay Description:
Inhibition of [3H]BRL-43694 binding to 5-hydroxytryptamine 3 receptor of rat cortical homogenate.
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
5-hydroxytryptamine receptor 3A
(GUINEA PIG)
European Research Centre For Drug Discovery And Development (Natsyndrugs)
Curated by
ChEMBL
Ligand
BDBM50060685
(9-Fluoro-4-(4-methyl-piperazin-1-yl)-pyrrolo[1,2-a...)
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Affinity Data
Kd: 64.6nM
Assay Description:
Antagonist activity at 5HT3 receptor in spontaneously beating guinea pig right atrium assessed as inhibition of serotonin-induced maximum response by...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI