Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAlpha-2A adrenergic receptor(BOVINE)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL

LigandBDBM50002154(5-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)Copy SMILESCopy InChI

Affinity DataKi:  270nMAssay Description:Binding affinity at Alpha-2 adrenergic receptor in calf cerebral cortex homogenates by [3H]clonidine displacement.More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetBeta-1 adrenergic receptor(GUINEA PIG)
Merck Sharp And Dohme Research Laboratories

Curated by ChEMBL

LigandBDBM50002154(5-Bromo-8-(4-methyl-piperazin-1-yl)-imidazo[1,2-a]...)Copy SMILESCopy InChI

Affinity DataKi:  500nMAssay Description:Binding affinity at Beta-1 adrenergic receptor in guinea pigs by [125I]CYP displacementMore data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/TrEMBL
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI