Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 6 hits in this display
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
IC50: 7nMAssay Description:All Examples were tested in HDAC1, 2, 3, 6 and 8 in vitro enzymatic assays. The assay principle is well known (Hauser et al. 2009, Bradner et al. 201...More data for this Ligand-Target Pair
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
IC50: 250nMAssay Description:All Examples were tested in HDAC1, 2, 3, 6 and 8 in vitro enzymatic assays. The assay principle is well known (Hauser et al. 2009, Bradner et al. 201...More data for this Ligand-Target Pair
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
IC50: 700nMAssay Description:All Examples were tested in HDAC1, 2, 3, 6 and 8 in vitro enzymatic assays. The assay principle is well known (Hauser et al. 2009, Bradner et al. 201...More data for this Ligand-Target Pair
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
IC50: 1.80E+3nMAssay Description:All Examples were tested in HDAC1, 2, 3, 6 and 8 in vitro enzymatic assays. The assay principle is well known (Hauser et al. 2009, Bradner et al. 201...More data for this Ligand-Target Pair
BDBM425889(N-hydroxy-2-{4-[(4- methylpiperazin-1- yl)methyl]p...)
IC50: 7.80E+3nMAssay Description:All Examples were tested in HDAC1, 2, 3, 6 and 8 in vitro enzymatic assays. The assay principle is well known (Hauser et al. 2009, Bradner et al. 201...More data for this Ligand-Target Pair