Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 15 hits in this display
IC50: 850nMAssay Description:Inhibition of GST-tagged BRD4 bromodomain (unknown origin) using biotinylated histone H4KAc peptide (1 to 21 residues) as substrate by HTRF assayMore data for this Ligand-Target Pair
IC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged BRD2 bromodomain-1 (65 to 187 residues) expressed in Escherichia coli expression system after 1...More data for this Ligand-Target Pair
IC50: >1.00E+5nMAssay Description:Inhibition of recombinant human N-terminal GST-tagged BRD3 bromodomain-2 (306 to 417 residues) expressed in Escherichia coli expression system after ...More data for this Ligand-Target Pair