Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 10 hits in this display
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: 129nMAssay Description:In vitro binding affinity at human recombinant 5-hydroxytryptamine 1A receptor in mammalian cells using 3[H]8-OH-DPAT as the radioligandMore data for this Ligand-Target Pair
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: 490nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 4 receptor in guinea pig striatum using 3[H]GR-113808 as the radioligandMore data for this Ligand-Target Pair
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: <1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 1B receptor in rat striatal muscles using [125I](-)-iodocyanopindolol as the radioligandMore data for this Ligand-Target Pair
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: <1.00E+3nMAssay Description:In vitro binding affinity to 5-hydroxytryptamine 2 receptor of rat cerebral cortex membranes using [3H]ketanserin as the radioligandMore data for this Ligand-Target Pair
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: <1.00E+3nMAssay Description:In vitro binding affinity at human recombinant 5-hydroxytryptamine 6 receptor in mammalian cells using 3[H]LSD as the radioligandMore data for this Ligand-Target Pair
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
BDBM50130276(CHEMBL553794 | N-Methyl-2-{2-[4-(2-oxo-1,2,4,5-tet...)
Ki: <1.00E+3nMAssay Description:In vitro binding affinity at 5-hydroxytryptamine 2C receptor in pig choroid plexus using 3[H]mesulergine as the radioligandMore data for this Ligand-Target Pair