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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetHistamine H4 receptor(Mus musculus (mouse))
Griffin Discoveries

Curated by ChEMBL
LigandPNGBDBM50433359(CHEMBL2376804)
Affinity DataKi:  15nMAssay Description:Binding affinity to mouse histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Rattus norvegicus (rat))
Griffin Discoveries

Curated by ChEMBL
LigandPNGBDBM50433359(CHEMBL2376804)
Affinity DataKi:  30nMAssay Description:Binding affinity to rat histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Griffin Discoveries

Curated by ChEMBL
LigandPNGBDBM50433359(CHEMBL2376804)
Affinity DataKi:  2.09E+4nMAssay Description:Displacement of [3H]histamine from human histamine H1 receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed