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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Histamine H4 receptor
(Homo sapiens (Human))
Argenta Discovery
Curated by
ChEMBL
Ligand
BDBM50315331
(1-(8-chlorobenzofuro[3,2-d]pyrimidin-4-yl)-N-methy...)
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Affinity Data
IC50: 76nM
Assay Description:
Inverse agonist activity at human histamine H4 receptor assessed as inhibition of [35S]GTPgammaS binding after 15 mins by scintillation proximity ass...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Histamine H4 receptor
(Homo sapiens (Human))
Argenta Discovery
Curated by
ChEMBL
Ligand
BDBM50315331
(1-(8-chlorobenzofuro[3,2-d]pyrimidin-4-yl)-N-methy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 87nM
Assay Description:
Displacement of [3H]histamine dihydrochloride from human histamine H4 receptor after 2.5 hrs by scintillation proximity assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI