Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetP2Y purinoceptor 1(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50409764(CHEMBL2112867)
Affinity DataKi:  3.60nMAssay Description:Inhibition of [3H]-5 binding to P2Y purinoceptor 1 expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2Y purinoceptor 1(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50409764(CHEMBL2112867)
Affinity DataIC50:  49nMAssay Description:Antagonistic activity against P2Y purinoceptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed