Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215404(CHEMBL227235 | [3-(2-iodo-6-methylaminopurin-9-yl)...)
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215404(CHEMBL227235 | [3-(2-iodo-6-methylaminopurin-9-yl)...)
IC50: 790nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215404(CHEMBL227235 | [3-(2-iodo-6-methylaminopurin-9-yl)...)
IC50: 794nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair