Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 3 hits in this display
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215400((1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(6-methy...)
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215400((1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(6-methy...)
IC50: 1.94E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeSADP-induced inositol phosphate formationMore data for this Ligand-Target Pair
P2Y purinoceptor 1(Homo sapiens (Human))National Institute Of Diabetes And Digestive And Kidney Diseases
Curated by ChEMBL
BDBM50215400((1'R,2'S,4'R,5'S)-phosphoric acid mono-[4-(6-methy...)
IC50: 1.95E+3nMAssay Description:Antagonist activity at human P2Y1 receptor expressed in 1321N1 cells assessed as inhibition of 2-MeS-ADP-stimulated PLC activityMore data for this Ligand-Target Pair