Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL

LigandBDBM50036668(CHEMBL3354799)Copy SMILESCopy InChI

Affinity DataEC50:  35nMAssay Description:Agonist activity at human GPR119 overexpressed in CHO cells assessed as increase in cellular cAMP production by HTRF methodMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Genomics Institute Of The Novartis Research Foundation

Curated by ChEMBL

LigandBDBM50036668(CHEMBL3354799)Copy SMILESCopy InChI

Affinity DataEC50:  15nMAssay Description:Agonist activity at human GPR119 overexpressed in CHO cells assessed as increase in cellular cAMP production by HTRF methodMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI