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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Mitogen-activated protein kinase kinase kinase 11
(Homo sapiens (Human))
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50108297
(CHEMBL288816 | Indolocarbazole analogue)
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Affinity Data
IC50: 31nM
Assay Description:
Inhibition of Mixed lineage kinase 3 (MLK3)
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mitogen-activated protein kinase kinase kinase 9
(Homo sapiens (Human))
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50108297
(CHEMBL288816 | Indolocarbazole analogue)
Copy SMILES
Copy InChI
Affinity Data
IC50: 45nM
Assay Description:
Inhibition of Mixed lineage kinase 1 (MLK1)
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mitogen-activated protein kinase kinase kinase 10
(Homo sapiens (Human))
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50108297
(CHEMBL288816 | Indolocarbazole analogue)
Copy SMILES
Copy InChI
Affinity Data
IC50: 89nM
Assay Description:
Inhibition of Mixed lineage kinase 2(MLK2)
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Protein kinase C alpha/beta/delta/epsilon/eta/gamma/theta/zeta type
(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50108297
(CHEMBL288816 | Indolocarbazole analogue)
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Copy InChI
Affinity Data
IC50: 980nM
Assay Description:
Binding affinity towards 5-hydroxytryptamine 3 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
High affinity nerve growth factor receptor
(Homo sapiens (Human))
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50108297
(CHEMBL288816 | Indolocarbazole analogue)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of NGF high affinity receptor tyrosine kinase TrkA
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI