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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  1.30nMAssay Description:Inhibition of serine protease factor Xa enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against Coagulation factor X in an enzyme inhibition assay.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  39nMAssay Description:Inhibition of serine protease trypsin enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  200nMAssay Description:Inhibition of serine protease thrombin enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  300nMAssay Description:Compound was tested for the inhibition of serine protease plasmin enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor VII(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  4.20E+3nMAssay Description:Compound was tested for the inhibition of serine protease factor VIIa enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50072448(CHEMBL18767 | {(3-Carbamimidoyl-phenyl)-[3-(2'-sul...)
Affinity DataKi:  3.30E+4nMAssay Description:Compound was tested for the inhibition of serine protease tissue plasminogen activator enzyme.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed