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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)

Curated by ChEMBL
LigandPNGBDBM50113255(5-[2-(5-Nitro-furan-2-yl)-vinyl]-furan-2-carboxyli...)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of GRK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetBeta-adrenergic receptor kinase 1(Homo sapiens (Human))
Centro De Investigaciones Biol�Gicas Margarita Salas (Csic)

Curated by ChEMBL
LigandPNGBDBM50113255(5-[2-(5-Nitro-furan-2-yl)-vinyl]-furan-2-carboxyli...)
Affinity DataIC50:  1.26E+5nMAssay Description:Inhibition of Beta-adrenergic receptor kinase 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed