Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetCREB-binding protein(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of CBP (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
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TargetHistone acetyltransferase p300(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of EP300 (unknown origin) by AlphaLISA immunodetection assayMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathway
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetHistone acetyltransferase KAT2B(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of PCAF (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of GCN5 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetHistone acetyltransferase KAT5(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of TIP60 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADantibodypediaGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetHistone acetyltransferase KAT7(Homo sapiens)
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MYST2 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBKEGG
UniProtKB/SwissProt
B.MOADGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI

TargetHistone acetyltransferase KAT6B(Homo sapiens)
Daiichi Sankyo

Curated by ChEMBL

LigandBDBM50579798(CHEMBL5080324)Copy SMILESCopy InChI

Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of MYST4 (unknown origin)More data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankGoogleScholar

Ligand InfoPC cidPC sid

In DepthDetails ArticlePubMed
Copy BDB DOI