Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Sepracor

Curated by ChEMBL
LigandPNGBDBM50301927(CHEMBL1748 | Norcisapride)
Affinity DataIC50:  19nMAssay Description:Displacement of [3H]GR-113808 from human recombinant 5-HT4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Sepracor

Curated by ChEMBL
LigandPNGBDBM50301927(CHEMBL1748 | Norcisapride)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H]granisetron from human recombinant 5-HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Sepracor

Curated by ChEMBL
LigandPNGBDBM50301927(CHEMBL1748 | Norcisapride)
Affinity DataEC50:  290nMAssay Description:Agonist activity at human recombinant 5-HT4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Sepracor

Curated by ChEMBL
LigandPNGBDBM50301927(CHEMBL1748 | Norcisapride)
Affinity DataEC50:  2.30E+3nMAssay Description:Antagonist activity at human recombinant 5-HT3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed