Home
About
Info
Download
WebServices
Contact
Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Sepracor
Curated by
ChEMBL
Ligand
BDBM50301927
(CHEMBL1748 | Norcisapride)
Copy SMILES
Copy InChI
Affinity Data
IC50: 19nM
Assay Description:
Displacement of [3H]GR-113808 from human recombinant 5-HT4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Sepracor
Curated by
ChEMBL
Ligand
BDBM50301927
(CHEMBL1748 | Norcisapride)
Copy SMILES
Copy InChI
Affinity Data
IC50: 1.60E+3nM
Assay Description:
Displacement of [3H]granisetron from human recombinant 5-HT3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 4
(Homo sapiens (Human))
Sepracor
Curated by
ChEMBL
Ligand
BDBM50301927
(CHEMBL1748 | Norcisapride)
Copy SMILES
Copy InChI
Affinity Data
EC50: 290nM
Assay Description:
Agonist activity at human recombinant 5-HT4 receptor
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
5-hydroxytryptamine receptor 3A
(Homo sapiens (Human))
Sepracor
Curated by
ChEMBL
Ligand
BDBM50301927
(CHEMBL1748 | Norcisapride)
Copy SMILES
Copy InChI
Affinity Data
EC50: 2.30E+3nM
Assay Description:
Antagonist activity at human recombinant 5-HT3 receptor expressed in HEK293 cells
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
Purchase
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI